Bioorganic & medicinal chemistry
Journal
Overview
publication venue for
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Di-indenopyridines as topoisomerase II-selective anticancer agents: Design, synthesis, and structure-activity relationships..
91.
2023
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Synthesis and biological evaluation of imidamide analogs as selective anti-trypanosomal agents..
61.
2022
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Dimeric small molecule agonists of EphA2 receptor inhibit glioblastoma cell growth..
28.
2020
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Lead optimization of selective tubulin inhibitors as anti-trypanosomal agents..
27.
2019
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Design, synthesis, and biological activity of substituted 2-amino-5-oxo-5H-chromeno[2,3-b]pyridine-3-carboxylic acid derivatives as inhibitors of the inflammatory kinases TBK1 and IKKε for the treatment of obesity..
26.
2018
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5-Adamantan thiadiazole-based thiazolidinones as antimicrobial agents. Design, synthesis, molecular docking and evaluation..
26.
2018
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Tetrahydroprotoberberine alkaloids with dopamine and σ receptor affinity..
24.
2016
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Development of a fluorescent cardiomyocyte specific binding probe..
24.
2016
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Ultrasmall dual-modality silica nanoparticle drug conjugates: Design, synthesis, and characterization..
23.
2015
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Design, synthesis, and immunologic evaluation of vaccine adjuvant conjugates based on QS-21 and tucaresol..
22.
2014
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Structure-guided design and development of novel benzimidazole class of compounds targeting DNA gyraseB enzyme of Staphylococcus aureus..
22.
2014
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Synthesis and biological evaluation of 18F-labled 2-phenylindole derivatives as PET imaging probes for β-amyloid plaques..
21.
2013
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Radiosynthesis of the tumor hypoxia marker [18F]TFMISO via O-[18F]trifluoroethylation reveals a striking difference between trifluoroethyl tosylate and iodide in regiochemical reactivity toward oxygen nucleophiles..
19.
2011
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Synthesis and serotonin transporter activity of 1,3-bis(aryl)-2-nitro-1-propenes as a new class of anticancer agents..
19.
2010
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Synthesis and in vitro toxicity of 4-MTA, its characteristic clandestine synthesis byproducts and related sulfur substituted alpha-alkylthioamphetamines..
18.
2010
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A kit method for the high level synthesis of [211At]MABG..
15.
2007
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Optimized design and synthesis of chemical dimerizer substrates for detection of glycosynthase activity via chemical complementation..
14.
2006
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Design, synthesis and biological evaluation of novel riccardiphenol analogs..
13.
2005
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A novel neoglycopeptide building block..
11.
2003
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Development of a purine-scaffold novel class of Hsp90 binders that inhibit the proliferation of cancer cells and induce the degradation of Her2 tyrosine kinase..
10.
2002
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Synthetic mannosides act as acceptors for mycobacterial alpha1-6 mannosyltransferase..
9.
2001
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Stereochemical influence on the stability of radio-metal complexes in vivo. Synthesis and evaluation of the four stereoisomers of 2-(p-nitrobenzyl)-trans-CyDTPA..
5.
1997
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Retinoic acid signaling pathways in development and diseases.
2013
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